FX-909

Based on 1 reference(s) in Google Scholar 8 10 1

Axon 4267

CAS [2924573-90-8]

MF C17H10F2N2O3S
MW 360.34

  • Purity: 98%
  • Soluble in DMSO

FX-909

Description

FX-909 is a first-in-class, orally available and highly potent covalent inverse agonist of the peroxisome proliferator-activated receptor gamma (PPARG) lineage transcription factor with cellular IC50 = 1 nM, highly selective over PPARA/PPARD (related transcription factors) (over 2000-fold selectivity).

KEYWORDS: FX-909 | Supplier | PPARG inverse agonist | FX909 | FX 909 | CT-FX909 | CAS [2924573-90-8] | PPAR-γ | Antagonist | Transcription Factors

Peroxisome proliferator-activated receptor gamma (PPARG) inverse agonist

Chemical name

3-(5,7-Difluoro-4-oxo-1,4-dihydroquinolin-2-yl)-4-(methylsulfonyl)benzonitrile

Source information

Sold in collaboration with Chemietek

Parent CAS No.

[2924573-90-8]

The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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