MR-2088

Based on 1 reference(s) in Google Scholar 8 10 1

Axon 4177

CAS [2922531-69-7]

MF C19H17F3N4OS
MW 406.43

  • Purity: 99%
  • Soluble in 0.1N HCl(aq), DMSO and EtOH
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MR-2088

Description

MR-2088 is a best-in-class, potent and selective ULK1/2 inhibitor with a ULK1 binding/activity of 2 nM. MR-2088 blocks autophagy flux and synergizes with Trametinib (Axon 1761) to provide antiproliferative effects in NSCLC.

KEYWORDS: MR-2088 | Supplier | ULK1/2 inhibitor | MR2088 | MR 2088 | CAS [2922531-69-7] | Non Selective (Phosphorylation substrates) | ULK | ULK1 | ULK2 | Inhibitor | Enzymes | Autophagy | UNC-51-like kinase

Best-in-class, potent and selective ULK1/2 inhibitor

Chemical name

4-(2-(1,2,5,6-Tetrahydropyridin-3-yl)-1H-pyrrolo[2,3-b]pyridin-5-yl)-N-(2,2,2-trifluoroethyl)thiophene-2-carboxamide

Parent CAS No.

[2922531-69-7]

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Size Unit Price Stock
5 mg €160.00 In Stock
25 mg €640.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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