GRL018-21

Based on 1 reference(s) in Google Scholar 8 10 1

Axon 4158

CAS [3061801-07-5]

MF C30H25FN4O5
MW 540.54

  • Purity: 98%
  • Optical purity: 100% e.e.
  • Soluble in DMSO
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GRL018-21

Description

GRL018-21 is a potent, highly selective and non-covalent GRK5 inhibitor with an IC50 value of 10 nM.

KEYWORDS: GRL018-21 | Supplier | GRK5 inhibitor | GRL 018-21 | GRL-018-21 | CAS [3061801-07-5] | Non Selective (Phosphorylation substrates) | GRK | Inhibitor | Enzymes | Chronic heart failure | G protein-coupled receptor kinase 5

Potent, highly selective and non-covalent GRK5 inhibitor

Chemical name

(R,Z)-N-(1-(4-Fluorophenyl)ethyl)-3-((4-(2-(furan-2-yl)-2-oxoacetamido)-3,5-dimethyl-1H-pyrrol-2-yl)methylene)-2-oxoindoline-5-carboxamide

Parent CAS No.

[3061801-07-5]

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Size Unit Price Stock
5 mg €180.00 In Stock
25 mg €720.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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