EPZ005687 hydrochloride - EPZ015938 hydrochloride

Based on 25 reference(s) in Google Scholar 8 10 25

Axon 4137

CAS [N.A.]

MF C32H37N5O3.HCl
MW 576.13

  • Purity: 99%
  • Soluble in DMSO
Recently added

EPZ005687 hydrochloride


EPZ005687 is a potent and selective small molecule inhibitor of histone methyltransferase EZH2 ( Ki = 24 nM). It has greater than 500-fold selectivity against 15 other protein methyltransferases and has 50-fold selectivity against the closely related enzyme EZH1.

Keywords: EPZ005687 hydrochloride | Supplier | EZH2 HMTase inhibitor | EPZ015938 hydrochloride | EPZ-005687 | EPZ 005687 | EPZ-015938 | EPZ 015938 | CT-EPZ687 | CAS [N.A.] | [1396772-26-1] | Histone | HMTase | Inhibitor | Enzymes

EZH2 HMTase inhibitor

Chemical name

1-Cyclopentyl-N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-6-(4-(morpholinomethyl)phenyl)-1H-indazole-4-carboxamide hydrochloride

Source information

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Parent CAS No.


The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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