Your cart

There are no items in your shopping cart

EPZ005687 hydrochloride - EPZ015938 hydrochloride

Based on 25 reference(s) in Google Scholar 8 10 25

Axon 4137

CAS [N.A.]

MF C32H37N5O3.HCl
MW 576.13

  • Purity: 99%
  • Soluble in DMSO

EPZ005687 hydrochloride

Description

EPZ005687 is a potent and selective small molecule inhibitor of histone methyltransferase EZH2 ( Ki = 24 nM). It has greater than 500-fold selectivity against 15 other protein methyltransferases and has 50-fold selectivity against the closely related enzyme EZH1.

Keywords: EPZ005687 hydrochloride | Supplier | EZH2 HMTase inhibitor | EPZ015938 hydrochloride | EPZ-005687 | EPZ 005687 | EPZ-015938 | EPZ 015938 | CT-EPZ687 | CAS [N.A.] | [1396772-26-1] | Histone | HMTase | Inhibitor | Enzymes

EZH2 HMTase inhibitor

Chemical name

1-Cyclopentyl-N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-6-(4-(morpholinomethyl)phenyl)-1H-indazole-4-carboxamide hydrochloride

Source information

Sold in collaboration with Chemietek

Parent CAS No.

[1396772-26-1]

Related Products

Axon ID Name Description From price
2140 GSK 126 Inhibitor of Histone Lysine Methyltransferase EZH2 €75.00
2227 EPZ 6438 Inhibitor of Histone Lysine Methyltransferase EZH2 €90.00
2701 EED226 Potent, selective and orally bioavailable PRC2 inhibitor €90.00
3469 MS1943 trifluoroacetate First-in-class EZH2 selective degrader; PROTAC €200.00
3695 PF-06821497 Inhibitor of Histone Lysine Methyltransferase EZH2 €160.00
3722 Valemetostat Inhibitor of Histone Lysine Methyltransferase EZH1/2 €160.00
4216 EPZ011989 hydrochloride Cell permeable, metabolically stable and orally available EZH2 inhibitor Inquire

The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

Newsletter
Give Feedback
 
Send E-mail

Customer Support

About Axon Medchem

Download Product Catalog

Download the Axon Ligands™ catalogue 2021 Spring Edition

Follow Us

© 2016 Axon Medchem. All Rights Reserved.

Send us a message

×

Contact Us

* Required Fields

Please wait...