Based on 17 reference(s) in Google Scholar 8 10 17

Axon 4136

CAS [1229652-21-4]

MW 463.29

  • Purity: 99%
  • Soluble in DMSO



HA130 is a potent and selective Autotaxin inhibitor (IC50 = 28 nM), binding and inhibiting Autotaxin reversibly. Displays no activity against the proteasome, recombinant NPP1 or alkaline phosphatase. Inhibits ATX-mediated cell migration in an A2058 melanoma cell assay.

Keywords: HA130 | Supplier | ATX inhibitor | HA-130 | HA 130 | CT-HA130 | CAS [1229652-21-4] | LPC | PDE | Inhibitor | Enzymes

Autotaxin (ATX) inhibitor

Chemical name

B-[3-[[4-[[3-[(4-Fluorophenyl)methyl]-2,4-dioxo-5-thiazolidinylidene]methyl]phenoxy]methyl]phenyl]-boronic acid,

Source information

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Parent CAS No.


The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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