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Enzymes
Hydrolases
Esterases (Phosphodi-)
PDE
ENPP1 inhibitor compound 43

ENPP1 inhibitor compound 43

Based on 1 reference(s) in Google Scholar 8 10 1

Axon 4042

CAS [2631703-41-6]

MF C16H18N6O3S
MW 374.42

Purity: 99%
Soluble in 0.1N NaOH(aq), 0.1N HCl(aq), DMSO and EtOH

ENPP1 inhibitor compound 43

Description

ENPP1 inhibitor compound 43 is a potent, selective and orally bioavailable ENPP1 inhibitor with a Ki value of 41 nM.

Keywords: ENPP1 inhibitor compound 43 | Supplier | ENPP1 inhibitor | CAS [2631703-41-6] | Cyclic 2'3'- cGAMP | PDE | Inhibitor | Enzymes | Cancer immunotherapy | Immune checkpoint inhibitor | Immune-oncology | Lung cancer | STING | Innate immunity | Ecto-nucleotide pyrophosphatase/phosphodiesterase 1 | NPP1

M Gangar et al. Design, synthesis and biological evaluation studies of novel small molecule ENPP1 inhibitors for cancer immunotherapy. Bioorg Chem. 2022 Feb;119:105549.

Cell Signaling & Oncology Immunology PDE EC 3.1.4.1

Potent, selective and orally bioavailable ENPP1 inhibitor

Chemical name

2-(2-Amino-7H-purin-6-ylthio)-N-(4-hydroxy-3-methoxyphenyl)butanamide

Parent CAS No.

[2631703-41-6]

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Size	Unit Price	Stock
10 mg	€220.00	In Stock
50 mg	€800.00	In Stock

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