GDC-0068 - Ipatasertib | RG7440

Based on 185 reference(s) in Google Scholar 8 10 185

Axon 4037

CAS [1001264-89-6]

MF C24H32ClN5O2
MW 458.00

  • Purity: 99%
  • Optical purity: 99% d.e.
  • Soluble in DMSO

GDC-0068

Description

GDC-0068 is a potent, APT-competitive and orally available small molecule pan-Akt inhibitor with IC50s of 5, 18 and 8 nM for Akt1, Akt2 and Akt3, respectively, and with selectivity over more than other 200 screened kinases. It displays robust antitumor activity with activation of PI3K-Akt-mTOR pathway.

KEYWORDS: GDC-0068 | Supplier | Akt inhibitor | Ipatasertib | RG7440 | GDC0068 | GDC 0068 | RG-7440 | RG 7440 | CT-G0068 | CAS [1001264-89-6] | Phosphatidylinositol | Akt | Inhibitor | Enzymes

Potent, APT-competitive and orally available small molecule pan-Akt inhibitor.

Chemical name

(S)-2-(4-Chlorophenyl)-1-(4-((5R,7R)-7-hydroxy-5-methyl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)piperazin-1-yl)-3-(isopropylamino)propan-1-one

Source information

Sold in collaboration with Chemietek

Parent CAS No.

[1001264-89-6]

The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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