BI-87G3 - NPAS3 heterodimer inhibitor compound 6

Based on 2 reference(s) in Google Scholar 8 10 2

Axon 4028

CAS [2207-44-5]

MF C10H5N3O2S3
MW 295.36

  • Purity: 98%
  • Soluble in DMSO

BI-87G3

Description

BI-87G3 is a highly potent covalent NPAS3 heterodimer inhibitor with a biochemical EC50 value of 282 nM. BI-87G3 effectively down-regulated NPAS3's transcriptional function by disrupting the interface of NPAS3-ARNT complexes at cellular level.

Keywords: BI-87G3 | Supplier | NPAS3 inhibitor | NPAS3 heterodimer inhibitor compound 6 | BI87G3 | BI 87G3 | CAS [2207-44-5] | DNA-RNA | PER-ARNT-SIM | Inhibitor | Transcription Factors | Neuronal regeneration | Neuronal development | Neuronal PAS domain protein 3 | Basic helix-loop-helix PER-ARNT-SIM | bHLH-PAS

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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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