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Enzymes
EC 2.3.2.13
LDN-27219

LDN-27219

Based on 3 reference(s) in Google Scholar 8 10 3

Axon 4016

CAS [312946-37-5]

MF C20H16N4O2S2
MW 408.50

Purity: 99%
Soluble in DMSO

LDN-27219

Description

LDN-27219 is a potent, reversible and slow-binding inhibitor of tissue transglutaminase (TGase) with an IC50 value of 0.6 μM.

Keywords: LDN-27219 | Supplier | TGase inhibitor | LDN27219 | LDN 27219 | CAS [312946-37-5] | Glutamine | Tgase | Inhibitor | Enzymes | Neurodegenerative disease

A Case et al. Kinetic analysis of the interaction of tissue transglutaminase with a nonpeptidic slow-binding inhibitor. Biochemistry. 2007 Jan 30;46(4):1106-15.

CNS EC 2.3.2.13

Potent, reversible and slow-binding TGase inhibitor

Chemical name

2-(4-Oxo-3,5-diphenyl-3,4-dihydrothieno[2,3-d]pyrimidin-2-ylthio)acetohydrazide

Parent CAS No.

[312946-37-5]

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Size	Unit Price	Stock
10 mg	€120.00	In Stock
50 mg	€480.00	In Stock

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