PF-03758309 - PF-3758309

Based on 42 reference(s) in Google Scholar 8 10 42

Axon 3961

CAS [N.A.]

MF C25H30N8OS.2HCl
MW 563.55

  • Purity: 99%
  • Optical purity: 99% e.e.
  • Soluble in water and DMSO

PF-03758309

Description

PF-03758309 is a potent, orally bioavailable and ATP-competitive inhibitor of p21-activated kinase (PAK), a downstream effector of the Rho family functioning as a signaling node for various oncogenic pathways.

KEYWORDS: PF-03758309 | Supplier | PAK4 Inhibitor | PF-3758309 | PF03758309 | PF 03758309 | PF3758309 | PF 3758309 | CT-PF0375 | CAS [N.A.] | [898044-15-0] | Non Selective (Phosphorylation substrates) | PAK | Inhibitor | Enzymes

Potent and ATP-competitive inhibitor of p21-activated kinase (PAK4)

Chemical name

(S)-N-(2-(Dimethylamino)-1-phenylethyl)-6,6-dimethyl-3-(2-methylthieno[3,2-d]pyrimidin-4-ylamino)-4,6-dihydropyrrolo[3,4-c]pyrazole-5(1H)-carboxamide

Source information

Sold in collaboration with Chemietek

Parent CAS No.

[898044-15-0]

The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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