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JG-2016

Based on 1 reference(s) in Google Scholar 8 10 1

Axon 3959

CAS [2887480-87-5]

MF C18H21ClN4O3
MW 376.84

  • Purity: 99%
  • Soluble in DMSO and EtOH

JG-2016

Description

JG-2016 is the first inhibitor of the HAT1 enzyme complex with an IC50 value of 14.8 μM. JG-2016 showed relative specificity toward HAT1 compared to other acetyltransferases, suppressed the growth of human cancer cell lines, impaired enzymatic activity in cellulo, and interfered with tumor growth.

Keywords: JG-2016 | Supplier | HAT1 inhibitor | JG 2016 | JG2016 | CAS [2887480-87-5] | Histone | HAT | Inhibitor | Enzymes

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Size Unit Price Stock
5 mg €140.00 In Stock
25 mg €560.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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