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Axon 3931

CAS [1022958-60-6]

MF C28H35ClN6O3
MW 539.07

  • Purity: 99%
  • Optical purity: 99%
  • Soluble in 0.1N HCl(aq) and DMSO



CEP-28122 is a highly potent, selective and orally active ALK inhibitor (Ezymatic IC50: 1.9 nM, 3 nM, Cellular IC50: 30 nM), Cellular IC50 in 75% murine: 300 nM), displaying a favorable pharmaceutical and pharmacokinetic profile and robust and selective pharmacologic efficacy against ALK-positive human cancer cells and tumor xenograft models in mice.

KEYWORDS: CEP-28122 | Supplier | ALK inhibitor | CEP28122 | CEP 28122 | CT-CEP281 | CAS [1022958-60-6] |  | Non Selective | ALK | Inhibitor | Enzymes

Highly potent, selective and orally active ALK inhibitor

Chemical name


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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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