Roluperidone - CYR101 | MT210 | MIN101

Based on 15 reference(s) in Google Scholar 8 10 15

Axon 3859

CAS [359625-79-9]

MF C22H23FN2O2
MW 366.43

  • Purity: 98%
  • Soluble in 0.1N HCl(aq) and DMSO

Roluperidone

Description

Roluperidone is a sigma-2 and 5-HT2A receptor antagonist with Ki values of 8.19 nM and 7.53 nM, respectively. Also, Roluperidone shows binding affinity for a1-adrenergic receptors but low or no affinity for muscarinic, cholinergic, and histaminergic receptors.

KEYWORDS: Roluperidone | Supplier | Sigma-2/5-HT2A antagonist | CYR101 | MT210 | MIN101 | CYR 101 | CYR-101 | MT 210 | MT-210 | MIN 101 | CAS [359625-79-9] | [359625-80-2] | [1937215-88-7] | Sigma receptor substrates | Sigma-2 | Antagonist | Receptors | Schizophrenia

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10 mg €120.00 In Stock
50 mg €420.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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