Your cart

There are no items in your shopping cart

GDC-1971 - RLY-1971

Based on 2 reference(s) in Google Scholar 8 10 2

Axon 3767

CAS [2377352-49-1]

MF C25H26N8O
MW 454.53

  • Purity: 99%
  • Optical purity: 98%
  • Soluble in DMSO and 0.1N HCl(aq)

GDC-1971

Description

GDC-1971 is an orally available, potent, and selective inhibitor of the protein tyrosine phosphatase SHP2, binding and stabilizing SHP2 in its inactive conformation.

KEYWORDS: GDC-1971 | Supplier | SHP2 inhibitor | RLY-1971 | GDC1971 | GDC 1971 | RLY1971 | RLY 1971 | CT-G1971 | CAS [2377352-49-1] | Non Selective (Tyrosine specific phosphomonoesters) | SHP | Inhibitor | Enzymes

Orally available, potent, and selective inhibitor of the protein tyrosine phosphatase SHP2

Chemical name

(R)-1'-(3-(3,4-dihydro-1,5-naphthyridin-1(2H)-yl)-1H-pyrazolo[3,4-b]pyrazin-6-yl)-3H-spiro[benzofuran-2,4'-piperidin]-3-amine

Source information

Sold in collaboration with Chemietek

Parent CAS No.

[2377352-49-1]

Related Products

Axon ID Name Description From price
2633 SHP099 Highly potent, selective and orally bioavailable SHP2 inhibitor €80.00
2723 TPI-1 Selective SHP1 inhibitor €95.00
3721 JAB-3068 SHP2 inhibitor €240.00
3865 TNO155 Selective and orally bioavailable allosteric inhibitor of SHP2 Inquire
3868 RMC-4550 hydrochloride Potent, selective and orally available small molecule allosteric inhibitor of SHP2 Inquire
3903 IACS-13909 hydrochloride Potent and specific allosteric inhibitor of SHP2 Inquire

The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

Newsletter
Give Feedback
 
Send E-mail

Customer Support

About Axon Medchem

Download Product Catalog

Download the Axon Ligands™ catalogue 2021 Spring Edition

Follow Us

© 2016 Axon Medchem. All Rights Reserved.

Send us a message

×

Contact Us

* Required Fields

Please wait...