KB-0742 dihydrochloride

Based on 2 reference(s) in Google Scholar 8 10 2

Axon 3730

CAS [2416874-75-2]

MF C16H25N5.2HCl
MW 360.33

  • Purity: 99%
  • Optical purity: 99% e.e.
  • Soluble in water
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KB-0742 dihydrochloride

Description

KB-0742 is an orally bioavailable, potent and selective CDK9 inhibitor with an IC50 of 6 nM, highly selective against other CDKs (>60 fold). Demonstrates in vitro and in vivo anti-tumor activity.

* Sold in collaboration with Chemietek.

KEYWORDS: KB-0742 dihydrochloride | Supplier | CDK9 inhibitor  | CT-KB0742 | CAS [2416874-75-2] | [2416873-83-9] | DNA-RNA | CDK9 | Inhibitor | Enzymes

Orally bioavailable, potent and selective CDK9 inhibitor

Chemical name

(1S,3S)-N1-(5-(pentan-3-yl)pyrazolo[1,5-a]pyrimidin-7-yl)cyclopentane-1,3-diamine dihydrochloride

Source information

Sold in collaboration with Chemietek

Parent CAS No.

[2416873-83-9]

The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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