PF-06939999 dihydrochloride

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Axon 3692

CAS [N.A.]

MF C22H23F3N4O3.2HCl
MW 521.36

  • Purity: 99%
  • Optical purity: 99% e.e.
  • Soluble in DMSO

PF-06939999 dihydrochloride

Description

PF-06939999  is an orally available and SAM competitive PRMT5 inhibitor binding to PRMT5-MEP-50 with high selectivity and affinity.

KEYWORDS: PF-06939999 dihydrochloride | PRMT5 inhibitor | PF06939999 | PF 06939999 | CT-PF0693 | CAS [N.A.] | [2159123-14-3] | Non Selective (Arginine Sites Proteins) | PRMT | Inhibitor | Enzymes

SAM competitive PRMT5 inhibitor

Chemical name

(1S,2S,3S,5R)-3-(6-(difluoromethyl)-5-fluoro-1,2,3,4-tetrahydroisoquinolin-8-yloxy)-5-(4-methyl-7H-pyrrolo[2,3-d]pyrimidin-7-yl)cyclopentane-1,2-diol

Source information

Sold in collaboration with Chemietek

Parent CAS No.

[2159123-14-3]

The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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