MS023 dihydrochloride

Based on 14 reference(s) in Google Scholar 8 10 14

Axon 3681

CAS [1992047-64-9]

MF C17H25N3O.2HCl
MW 360.32

  • Purity: 99%
  • Soluble in water, DMSO and EtOH
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MS023 dihydrochloride

Description

MS023 dihydrochloride is a potent, selective, and cell-active inhibitor of human Type I Protein Arginine Methyltransferases (IC50 values 30 nM, 119 nM, 83 nM, 4 nM, and 5 nM for PRMT1, PRMT3, PRMT4, PRMT6, and PRMT8, respectively) completely inactive against type II and type III PRMTs, protein lysine methyltransferases and DNA methyltransferases. MS023 potently decreased cellular levels of histone arginine asymmetric dimethylation.

KEYWORDS: MS023 dihydrochloride | Supplier | PRMT inhibitor | MS 023 dihydrochloride | MS-023 dihydrochloride | CAS [1992047-64-9] | [1831110-54-3] | [2117404-42-7] | [2108631-19-0] | Non Selective (Arginine Sites Proteins) | PRMT | Inhibitor | Enzymes

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5 mg €90.00 In Stock
25 mg €290.00 In Stock
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2 x 5 mg €140.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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