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GSK1278863 - Daprodustat

Based on 55 reference(s) in Google Scholar 8 10 55

Axon 3615

CAS [960539-70-2]

MF C19H27N3O6
MW 393.43

  • Purity: 99%
  • Soluble in 0.1N NaOH(aq), DMSO and EtOH
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GSK1278863

Description

GSK1278863 is a potent, selective and orally active inhibitor of all three HIF prolyl hydroxylase isozymes, PHD1, PHD2, and PHD3 with IC50 values of 3.5, 22.2 and 5.5 nM, respectively.

KEYWORDS: GSK1278863 | Supplier | HIF-PHD inhibitor | Daprodustat | GSK 1278863 | GSK-1278863 | CAS [960539-70-2] | Hypoxia-signaling cascade | PHD(HIF) | Inhibitor | Enzymes | Anemia | Chronic kidney disease

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Size Unit Price Stock
10 mg €120.00 In Stock
50 mg €420.00 In Stock
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Related Products

Axon ID Name Description From price
1921 IOX2 Inhibitor of Hypoxia Inducible Factor PHD €95.00
1948 HIF Phd Inhibitor 4 Inhibitor of Hypoxia Inducible Factor PHD €105.00
1977 DMOG Cell-permeable HIF-PHD inhibitor with pro-angiogenic and -osteogenic properties €65.00
2570 FG-2216 Orally active HIF-PHD inhibitor that increases plasma EPO levels in vivo €80.00
2588 FG-4592 New-generation oral HIF-PHD inhibitor €55.00
3095 MK-8617 Potent, orally active pan-inhibitor of HIF-PHD €90.00
3288 Vadadustat Oral HIF-PH inhibitor and HIF stabilizer €80.00

The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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