AMG510 - Sotorasib

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Axon 3575

CAS [2296729-00-3]

MF C30H30F2N6O3
MW 560.59

  • Purity: 99%
  • Optical purity: Optically pure
  • Soluble in DMSO

AMG510

Description

AMG510 is a highly potent, selective, orally bioavailable, well-tolerated and covalent KRASG12C inhibitor with an IC50 value of 68 nM (p-ERK).

KEYWORDS: AMG510 | Supplier | KRAS-G12C inhibitor | Sotorasib | AMG 510 | AMG-510 | CAS [2296729-00-3] | [2252403-56-6] | GTP | KRAS | Inhibitor | Enzymes | Lumakras | RAS

Highly potent, selective, and orally bioavailable KRAS-G12C inhibitor

Chemical name

4-((S)-4-Acryloyl-2-methylpiperazin-1-yl)-6-fluoro-7-(2-fluoro-6-hydroxyphenyl)-1-(2-isopropyl-4-methylpyridin-3-yl)pyrido[2,3-d]pyrimidin-2(1H)-one

Parent CAS No.

[2296729-00-3]

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Size Unit Price Stock
5 mg €90.00 In Stock
25 mg €300.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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