Based on 78 reference(s) in Google Scholar 8 10 78

Axon 3560

CAS [1604810-83-4]

MF C31H28ClN7O2
MW 566.05

  • Purity: 98%
  • Soluble in DMSO



THZ1 is a first covalent inhibitor of CDK7 (IC50 value of 3.2 nM) which employs a unique mechanism, combining ATP-site and allosteric covalent binding, as means of attaining potency and selectivity for CDK7. The dihydrochloride salt of THZ1 is also available as Axon 3561.

KEYWORDS: THZ1 | Supplier | CDK7 inhibitor | THZ 1 | THZ-1 | CAS [1604810-83-4] | [2422107-17-1] | Cyclin Dependent (CDK) | CDK | Inhibitor | Enzymes | T-cell acute lymphoblastic leukaemia | T-ALL | RUNX1

Size Unit Price Stock
2 mg €60.00 In Stock
5 mg €110.00 In Stock
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Size Unit Price Stock
2 x 5 mg €160.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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