BC-DXI-843

Based on 1 reference(s) in Google Scholar 8 10 1

Axon 3259

CAS [2421117-98-6]

MF C28H26N4O4S2
MW 546.66

  • Purity: 99%
  • Optical purity: 100% e.e.
  • Soluble in DMSO

BC-DXI-843

Description

BC-DXI-843 is a potent AIMP2-DX2 inhibitor (IC50 value of 0.92 μM) with more than 100-fold selectivity over AIMP2 in a luciferase assay. Moreover, BC-DXI-843 demonstrated in vivo efficacy in a tumor xenograft mouse model (H460 cells).

KEYWORDS: BC-DXI-843 | Supplier | AIMP2-DX2 inhibitor | BC-DXI843 | BC-DXI 843 | CAS [2421117-98-6] | Protein synthesis | Inhibitor | Proteins | Lung cancer | HSP70 | AIMP2 splicing variant | Ubiquitination | Aminoacyl-tRNA synthetase

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Size Unit Price Stock
10 mg €120.00 In Stock
50 mg €420.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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