GLPG1690 - Ziritaxestat

Based on 20 reference(s) in Google Scholar 80 100 20

Axon 3094

CAS [1628260-79-6]

MW 588.70

  • Purity: 98%
  • Soluble in DMSO



GLPG1690 is a first-in-class, potent autotaxin (ATX) inhibitor with a Ki value of 15 nM. GLPG1690 demonstrated significant activity in the mouse BLM-induced fibrosis model at doses of 10 and 30 mg/kg twice a day, with an efficacy comparable or superior to that of the reference compound pirfenidone.

KEYWORDS: GLPG1690 | supplier | ATX inhibitor | Ziritaxestat | GLPG 1690 | GLPG-1690 | CAS [1628260-79-6] | LPC | PDE | Inhibitor | Enzymes | Idiopathic pulmonary fibrosis

Size Unit Price Stock
10 mg €110.00 In Stock
50 mg €330.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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