BET BRD4 inhibitor compound II-25

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Axon 3037

CAS [1660117-38-3]

MF C25H27N5O2
MW 429.51

  • Purity: 99%
  • Optical purity: Optically pure
  • Soluble in 0.1N HCl(aq) and DMSO

BET BRD4 inhibitor compound II-25

Description

BET BRD4 inhibitor compound II-25 is a potent BRD4-BD1 inhibitor with an IC50 of 8 nM.

KEYWORDS: BET BRD4 inhibitor compound II-25 | BET inhibitor | BI 894999 | BI894999 | BI-894999 | CAS [1660117-38-3] | Histone | BET (BRD) | Inhibitor | Proteins | AML | Acute myeloid leukemia

Potent, selective and orally active BET inhibitor

Chemical name

(S)-2,4-Dimethyl-6-(1-(1-phenylethyl)-6-(tetrahydro-2H-pyran-4-yl)-1H-imidazo[4,5-c]pyridin-2-yl)pyridazin-3(2H)-one

Parent CAS No.

[1660117-38-3]

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5 mg €165.00 In Stock
25 mg €665.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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