A2764 dihydrochloride - TRESK inhibitor A2764

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Axon 3019

CAS [861038-72-4]

MF C15H19ClN2O.2HCl
MW 351.70

  • Purity: 99%
  • Soluble in water and DMSO
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A2764 dihydrochloride

Description

A2764 dihydrochloride is a selective inhibitor of TRESK (KCNK18) with an IC50 value of 11.8 μM. The degree of inhibition by 100 µM A2764 was larger in the activated state of TRESK than in the resting state of the channel. A2764 can inhibit TRESK in native cells, leading to cell depolarization and increased excitability.

KEYWORDS: A2764 dihydrochloride | supplier | TRESK inhibitor | A 2764 dihydrochloride | A-2764 dihydrochloride | CAS [861038-72-4] | [809248-52-0] | Potassium | TRESK | Inhibitor | Ion Channels | Migraine | Neuropathic pain | K2P18.1

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50 mg €305.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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