C 7280948

Based on 15 reference(s) in Google Scholar 8 10 15

Axon 2210

CAS [587850-67-7]

MF C14H16N2O2S
MW 276.35

  • Purity: 99%
  • Soluble in DMSO

C 7280948


Sulfone inhibitor of PRMT1 (IC50 values 12.75 μM and 26.7 μM for oligopeptide that contains the amino acids 1–21 of human histone H4 and non-histone protein Npl3 as methylation substrates respectively). Useful tool in studying the epigenetic role of PRMT1. PRMT1 has been linked to the activation of estrogen and androgen receptors as well. PRMT1 is a necessary component for oncogenic transformation induced by a mixed lineage leukemia (MLL) complex, and therefore may represent a new treatment option for hormone-dependent cancer.
Size Unit Price Stock
10 mg €85.00 In Stock
50 mg €255.00 In Stock
Special Offers
Size Unit Price Stock
2 x 10 mg €140.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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