TD 5108 - Velusetrag

Based on 20 reference(s) in Google Scholar 80 100 20

Axon 2060

CAS [866933-46-2]

MF C25H36N4O5S
MW 504.64

Purity: 99%
Optical purity: Optically pure
Soluble in 0.1N HCl(aq) and DMSO

TD 5108

Description

Potent and selective 5-HT4 receptor agonist with high intrinsic activity; drug candidate for the treatment of chronic constipation and irritable bowel syndrome

JAM Smith et al. The in vitro pharmacological profile of TD-5108, a selective 5-HT4 receptor agonist with high intrinsic activity. Naunyn-Schmiedeberg's Arch. Pharmacol. 2008, 378(1), 125-137.

ML Manini et al. Effects of Velusetrag (TD‐5108) on gastrointestinal transit and bowel function in health and pharmacokinetics in health and constipation. Neurogastroenterol. Motility, 2010, 22(1), 42-e8.

CNS 5-HT4 A19

Selective 5-HT4 receptor agonist

Chemical name

N-(8-((R)-2-hydroxy-3-(N-methylmethylsulfonamido)propyl)-8-azabicyclo[3.2.1]octan-3-yl)-1-isopropyl-2-oxo-1,2-dihydroquinoline-3-carboxamide

Parent CAS No.

[866933-46-2]

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