PF 04981517 - CYP3cide | PF 4981517

Based on 14 reference(s) in Google Scholar 8 10 14

Axon 2026

CAS [1390637-82-7]

MF C26H32N8
MW 456.59

  • Purity: 98%
  • Optical purity: Optically pure
  • Soluble in 0.1N HCl(aq) and DMSO

PF 04981517

Description

Potent and selective inhibitor of Cytochrome P450 3A4 (CYP3A4) with IC50 value of 30 nM; inactivates human CYP3A4 in an efficient and time-dependent manner
Inhibitor of Cytochrome P450 3A4 (CYP3A4)

Chemical name

(S)-1-methyl-3-(1-methyl-5-p-tolyl-1H-pyrazol-4-yl)-4-(3-(piperidin-1-yl)pyrrolidin-1-yl)-1H-pyrazolo[3,4-d]pyrimidine

Source information

Pfizer compound; Sold for research purposes under agreement from Pfizer Inc.

Parent CAS No.

[1390637-82-7]

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10 mg €110.00 In Stock
50 mg €380.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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