ERB 041 - Prinaberel

Based on 20 reference(s) in Google Scholar 80 100 20

Axon 1898

CAS [524684-52-4]

MF C15H10FNO3
MW 271.24

Purity: 99%
Soluble in 0.1N NaOH(aq) and DMSO

ERB 041

Description

Highly selective estrogen receptor β (ERβ) agonist, with IC50 value of 5.4 nM for human ERβ which is >200-fold selective over Erα

HA Harris et al. Evaluation of an estrogen receptor-beta agonist in animal models of human disease. Endocrinology 2003, 144(10), 4241-4249.

KF Koehler et al. Reflections on the discovery and significance of estrogen receptor beta. Endocr Rev. 2005, 26(3), 465-478.

XL Wang et al. ERB-041, a selective ER beta agonist, inhibits iNOS production in LPS-activated peritoneal macrophages of endometriosis via suppression of NF-kappaB activation. Mol. Immunol. 2009, 46(11-12), 2413-2418.

Selective estrogen receptor β (ERβ) agonist

Chemical name

2-(3-fluoro-4-hydroxyphenyl)-7-vinylbenzo[d]oxazol-5-ol

Parent CAS No.

[524684-52-4]

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10 mg	€95.00	In Stock
50 mg	€380.00	In Stock

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ERB 041 - Prinaberel

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ERB 041 - Prinaberel

Description

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