K+ Channel inhibitor 1734

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Axon 1734

CAS [343240-54-0]

MF C15H13Cl2N3O2
MW 338.19

  • Purity: 97%
  • Optical purity: racemate
  • Soluble in DMSO and Ethanol

K+ Channel inhibitor 1734

Description

Building block for synthesis of dihydropyrazolopyrimidine inhibitors of Kv1.5 (IKur). The ethylester analog of inhibitor 1734 is a modest inhibitor itself (IC50 value 1.1 µM for human Kv1.5), but exhibiting encouraging KV1.5 versus L-type calcium channel selectivity.

KEYWORDS: K+ Channel inhibitor 1734 | supplier | Building block | CAS [343240-54-0] | [1026960-80-4] | Potassium | Kv1.5 | Ikur | BMS | L-type | calcium channel 

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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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