CP 615003 mesylate

Based on 20 reference(s) in Google Scholar 80 100 20

Axon 1604

CAS [1259477-42-3]

MF C20H24FN3O3.CH4O3S
MW 469.53

Purity: 99%
Soluble in water and DMSO

CP 615003 mesylate

Description

A potent and subtype selective GABAA receptor partial agonist potentially useful in treating generalized anxiety disorder; the Mdr1 P-glycoprotein (P-gp) substrate

CL Shaffer et al. Metabolism and disposition of a g-aminobutyric acid type A receptor partial agonist in humans. Drug Metab. Disp. (2008), 36(4), 655-662.

K Venkatakrishnan et al. Central nervous system pharmacokinetics of the Mdr1 P-glycoprotein substrate CP-615,003. Drug Metab. Disp. (2007), 35(8), 1341-1349

GABAA agonist

Chemical name

N-(3-fluoro-4-(2-(propylamino)ethoxy)phenyl)-4-oxo-4,5,6,7-tetrahydro-1H-indole-3-carboxamide methanesulfonate

Parent CAS No.

[329016-45-7]

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5 mg	€90.00	In Stock
25 mg	€270.00	In Stock

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Size	Unit Price	Stock
2 x 5 mg	€140.00	In Stock
2 x 25 mg	€400.00	In Stock

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CP 615003 mesylate

Description

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Parent CAS No.

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CP 615003 mesylate

Description

Chemical name

Parent CAS No.

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