GSK 2126458 - Omipalisib

Based on 12 reference(s) in Google Scholar 9 10 12

Axon 1596

CAS [1086062-66-9]

MF C25H17F2N5O3S
MW 505.50

  • Purity: 99%
  • Soluble in DMSO

GSK 2126458

Description

Highly potent and orally bioavailable inhibitor of PI3K and mTOR in vitro and in vivo; Ki values to be 0.019, 0.13, 0.024 and 0.06 nM for p110 α, β, δ and γ isoforms and 0.18 and 0.3 nM for mTORC1 and mTORC2 respectively.

KEYWORDS: GSK 2126458 | supplier | PI3K/mTOR inhibitor | Omipalisib | GSK2126458 | GSK-2126458 | CAS [1086062-66-9] | Phosphatidylinositol | mTOR | PI3K | orally bioavailable | TORC

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Size Unit Price Stock
2 mg €80.00 In Stock
5 mg €120.00 In Stock
25 mg €420.00 In Stock
Special Offers
Size Unit Price Stock
2 x 5 mg €180.00 In Stock
2 x 25 mg €600.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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