Nalbuphine hydrochloride

Based on 20 reference(s) in Google Scholar 80 100 20

Axon 1577

CAS [23277-43-2]

MF C21H27NO4.HCl
MW 393.90

Purity: 99%
Soluble in water

Nalbuphine hydrochloride

Description

A narcotic used as a pain medication. Nalbuphine appears to be an agonist at κ-opioid receptors and an antagonist or partial agonist at μ-opioid receptors (IC50 of 36 nM and 11 nM resp).

P Gharagozlou et al. Activity of opioid ligands in cells expressing cloned µ opioid receptors. B.M.C. Pharmacol. 2003, 3, 1-8.

K Yasuda et al. Cloning and functional comparison of kappa and delta opioid receptors from mouse brain. Proc. Natl. Acad. Sci. USA. 1993, 90, 6736-6740.

Analgesic. Κ-opioid agonist and μ-opioid antagonist/partial agonist

Chemical name

(–)-17-(cyclobutylmethyl)- 4,5α-epoxymorphinan- 3,6α,14-triol Hydrochloride

Parent CAS No.

[20594-83-6 ]

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Nalbuphine hydrochloride

Description

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Nalbuphine hydrochloride

Description

Chemical name

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