GDC 0941 bismesylate - Pictilisib

Based on 190 publications in PubMed 10 10 190

Axon 1377

CAS [957054-33-0]

MF C23H27N7O3S2.2CH4O3S
MW 705.85

  • Purity: 99%
  • Soluble in water and DMSO

GDC 0941 bismesylate

Description

Potent, selective, orally bioavailable inhibitor of class I PI3 kinase (PI3K) under clinical trials, with IC50 values (nM) of 3, 33, 3, 75, 1230 and 580 for p110 α, β, δ and γ isoforms, DNA-PK and mTOR; water-soluble form.

KEYWORDS: GDC 0941 bismesylate | supplier | PI3K inhibitor | Pictilisib | GDC0941 | GDC-0941 | CAS [957054-33-0] | [957054-30-7] | Phosphatidylinositol | orally bioavailable | p110-alpha | DNA-PK | mTOR |  water-soluble

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5 mg €85.00 In Stock
25 mg €255.00 In Stock
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2 x 5 mg €120.00 In Stock
2 x 25 mg €360.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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