Axon LigandsTM for Drug Discovery
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[e-catalogue available in pdf]
Products - Axon Ligands TM - List of New Ligands (by date added) 2011 2010 2009 2008
(Back to New Ligands Released)
2011 DEC
(-)-Bay-K8644 | Ca chan. activator
(+)-Bay-K8644 | Ca chan. modulator
(S)-WAY100135 | 5-HT1A antag.
(R)-WAY100135 | 5-HT1A antag.
NXY 059 | radical scavenger
A 770041 | Lck inhibitor
EGFR inhibitor [879127-07-8]
Apixaban | Factor Xa inhibitor
dl-hCPT | Topo-1 inhibitor
ADL 5859 | δ opioid agonist
AZ 12216052 | mGluR8 PAM
PF 3845 | FAAH inhibitor
VU 0357017 | M1 PAM
MK 0354 | Naicin partial agonist
SEW 2871 | S1P1 agonist
BMS 345541 | IKK inhibitor
WAY 208466 | 5-HT6 agonist
SB 242084 | 5-HT2C antagonist
2011 NOV
PPP | CYP2B6 inhibitor
Brimonidine | α2 agonist
PAC-1 | Procaspase activator
AMD 3100 | CXCR4 antagonist
Kifunensine | Mannosidase inh.
Palomid 529 | Akt/mTOR inhibitor
Venlafaxine | SNRI
Bexarotene | RXR agonist
A 83-01 | ALK5 inhibitor
BI 6727 | PLK1 inhibitor
GB 83 | PAR2 antagonist
2011 OCT
GSK 690693 | AKT inhibitor
AC 220 | FLT3 inhibitor
SLV 319 | CB1 antagonist
BXL 628 | VDR agonist
Temsirolimus | mTOR inhibitor
REP 3123 | MetRS inhibitor
REP 8839 | MetRS inhibitor
Orvepitant | NK1 antagonist
FR 180204 | ERK inhibitor
BIO | GSK3 inhibitor
2011 SEP
OSI 906 | IGF-1R/IR inhibitor
Shz-1 | Differentiating agent
SU 5402 | FGFR inhibitor
BIX 01294 | HMTase inhibitor
RG 108 | DNA methylation inh.
YS 49 | antithrombotic
MDL 201012 | M3 antagonist
STF 083010 | IRE1 inhibitor
PF 02341066 | c-Met/ALK inh.
2011 AUG
KU 55933 | ATM inhibitor
LY 317615 | PKCβ inhibitor
GSK 461364 | PLK1 inhibitor
CYT 387 | JAK1/2 inhibitor
Asoprisnil | PR modulator
RU 58841 | Antiandrogen
AEE 788 | EGFR/VEGFR inhibitor
MK 2206 | AKT inhibitor
Y-27632 | ROCK inhibitor
2011 JULY
R 406 | Syk inhibitor
BAY 73-4506 | RTK inhibitor
BINA | mGluR2 PAM
Danoprevir | HCV protease inh.
PD 173074 | FGFR inhibitor
TWS 119 | GSK-3β inhibitor
SCIO 469 | p38 MAPK inhibitor
2011 JUN
PHA 408 | IKK-2 inhibitor
Digoxin | HIF-1 inhibitor
A 357300 | MetAP-2 inhibitor
LY 334370 | 5-HT1F agonist
Pelitinib | EGFR inhibitor
Reversine | Dedifferentiation agent
Perifosine | AKT inhibitor
CP 547632 | VEGFR2 inhibitor
2011 MAY
PS 47 | E-isomer of PS48
PS 48 | PDK1 activator
HLI 373 | HDM2 inhibitor
SB 431542 | ALK5 inhibitor
Thiazovivin | hESC enhancer
Irestatin 9389 | IRE1 inhibitor
S9947 | IKur channel blocker
2011 APR
CP 100356 | P-gp inhibitor
ISOX | HDAC6 inhibitor
MK 0364 | CB1 inverse agonist
Ambrisentan | ETA antagonist
YM 155 | Survivin suppresant
NN 414 | KATP channel opener
AZ 23 | Trk inhibitor
AZ 3146 | Mps1 inhibitor
2011 MAR
HTI 286 | Tubulin inhibitor
CHIR 124 | CHK1 inhibitor
Zaleplon | Benzodiazepine ago.
NSC 23766 | Rac1 inhibitor
CGP 57380 | MNK1 inhibitor
ABT 869 | RTK inhibitor
PF 573228 | FAK inhibitor
GSK 3787 | PPAR δ antagonist
VER 155008 | Hsp70 inhibitor
2011 FEB
Sotrastaurin | PKC inhibitor
CID 755673 | PKD inhibitor
XMD8-92 | BMK1 inhibitor
OSI 420 | EGFR inhibitor
Vildagliptin | DPP4 inhibitor
Ruxolitinib | JAK1/2 inh.
Remogliflozin | SGLT2 inhibitor
NVP-LDE225 | SMO antagonist
SGI 1776 | Pim inhibitor
2011 JAN
Aurora A inhibitor II | AurA inh.
GSK 461364 analog I | PLK1 inh.
GSK 461364 analog II | PLK1 inh.
Aurora A inhibitor I | AurA inh.
CDIBA | cPLA2 inhibitor
PF 4708671 | S6K1 inhibitor
SB 265610 | CXCR2 antagonist
SNS 032 | CDK 2 inhibitor
HMR 1031 | VLA-4 antagonist
NVP 231 | CerK inhibitor
CP 615003 | GABAA agonist
2012: NEW JAN; 2011: DEC NOV OCT SEP AUG JULY JUN MAY APR MAR FEB JAN; See 2011 2010 2009
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