Axon LigandsTM for Drug Discovery
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Brand-new like kinase inhibitors...
[e-catalogue available in pdf]
Products - Axon Ligands TM - List of New Ligands (by date added) 2011 2010 2009 2008
New Ligands Released:
A 784168 | TRPV1 antagonist
IMS 2186 | Apoptosis inducer
MS 275 | HDAC inhibitor
NVP-BHG712 | EphB4 inhibitor
AP 24534 | BCR-ABL inhibitor
VU 0364770 | mGuR4 PAM
VU 0361737 | mGuR4 PAM
Erastin | VDAC2 inhibitor
BH3I-1 | Bcl-xL antagonist
PF 04691052 | PI3K/mTOR inh.
ARQ 197 | MET inhibitor
A 66 | PI3K p110α inhibitor
Rolofylline M1-trans | A1 antag.
Rolofylline M1-cis | A1 antag.
PCI 34051 | HDAC8 inhibitor
Torin 1 | mTOR inhibitor
Torin 2 | mTOR inhibitor
DBeQ | p97 inhibitor
MK 0822 | Cathepsin K inhibitor
CK 1827452 | Myosin activator
Sulfonamide 13 | JAK2 inhibitor
Eeyarestatin 1 | ERAD inhibitor
CCT 137690 | Aurora inhibitor
UNC 0224 | HMTase inhibitor
GW 788388 | TGF-βR1 inhibitor
C646 | p300 HAT inhibitor
Wiskostatin | N-WASP inhibitor
N6022 | GSNOR inhibitor
XL PI3K/mTOR inh. | Axon 1706
PKI 587 | PI3K/mTOR inhibitor
2012 APR
BIX 02189 | MEK5/ERK5 inhibitor
Cabozantinib | MET/VEGFR2 inh.
GS 39783 | GABAB PAM
Pyroxamide | HDAC inhibitor
CCT007093 | PPM1D inhibitor
NQDI-1 | ASK1 inhibitor
S 18986 | AMPA PAM
PF 4800567 | CK 1e inhibitor
VU 0360223 | mGluR5 antagonist
NVP-BGJ398 | FGFR inhibitor
MC 1568 | IIa HDAC inhibitor
VX 745 | p38α MAPK inhibitor
BAN ORL 24 | NOP antagonist
JTC 801 | NOP antagonist
Bortezomib | Proteasome inhibitor
LB 42708 | FTase inhibitor
PDE5 inhibitor | Axon 1709
2012 MAR
(S)-3,5-DHPG | mGluR1 agonist
(RS)-3,5-DHPG | mGluR1 agonist
CXCR3 antagonist | Axon 1800
SCH 727965 | CDK inhibitor
Nav1.7 blocker | Axon 1780
Nav1.7 blocker | Axon 1791
VU 0255035 | M1 antagonist
GSK 2126458 | PI3K/mTOR inh.
BKM 120 | PI3K inhibitor
SC 66 | AKT inhibitor
CaSR antagonist | Axon 1732
FXR 450 | FXR inhibitor
Kv1.3 blocker | Axon 1735
AMG 900 | Aurora inhibitor
WP 1130 | DUB inhibitor
SB 939 | HDAC inhibitor
AMG 706 | VEGFR inhibitor
2012 FEB
GDC 0980 | PI3K/mTOR inhibitor
VU 0238429 | M5 PAM
MG 149 | Tip60 HAT inhibitor
AZ 960 | JAK2 inhibitor
SA 4503 | Sigma-1 agonist
TG 003 | Clk inhibitor
D-Atazanivir | Protease inhibitor
SCH 530348 | PAR1 antagonist
HMR 1098 | KATP chan. blocker
2012 JAN
Iobenguane | MIBG standard
PNU 100480 | Anti-TB agent
BVT 2733 | 11β-HSD1 inhibitor
Doxercalciferol | VDR agonist
CoPo-22 | CFTR CoPo
T 1776Na | PAI-1 inhibitor
GSK 1120212 | MEK inhibitor
CDDO-Me | Apoptosis inducer
ICG 001 | Wnt/CREB inhibitor
Bazedoxifene | SERM
2011 DEC
(-)-Bay-K8644 | Ca chan. activator
(+)-Bay-K8644 | Ca chan. modulator
(S)-WAY100135 | 5-HT1A antag.
(R)-WAY100135 | 5-HT1A antag.
NXY 059 | radical scavenger
A 770041 | Lck inhibitor
EGFR inhibitor [879127-07-8]
Apixaban | Factor Xa inhibitor
dl-hCPT | Topo-1 inhibitor
ADL 5859 | δ opioid agonist
AZ 12216052 | mGluR8 PAM
PF 3845 | FAAH inhibitor
VU 0357017 | M1 PAM
MK 0354 | Naicin partial agonist
SEW 2871 | S1P1 agonist
BMS 345541 | IKK inhibitor
WAY 208466 | 5-HT6 agonist
SB 242084 | 5-HT2C antagonist
2011 NOV
PPP | CYP2B6 inhibitor
Brimonidine | α2 agonist
PAC-1 | Procaspase activator
AMD 3100 | CXCR4 antagonist
Kifunensine | Mannosidase inh.
Palomid 529 | Akt/mTOR inhibitor
Venlafaxine | SNRI
Bexarotene | RXR agonist
A 83-01 | ALK5 inhibitor
BI 6727 | PLK1 inhibitor
GB 83 | PAR2 antagonist
2011 OCT
GSK 690693 | AKT inhibitor
AC 220 | FLT3 inhibitor
SLV 319 | CB1 antagonist
BXL 628 | VDR agonist
Temsirolimus | mTOR inhibitor
Bay K8644 | Ca chan. activator
REP 3123 | MetRS inhibitor
REP 8839 | MetRS inhibitor
Orvepitant | NK1 antagonist
FR 180204 | ERK inhibitor
BIO | GSK3 inhibitor
2011 SEP
OSI 906 | IGF-1R/IR inhibitor
Shz-1 | Differentiating agent
SU 5402 | FGFR inhibitor
BIX 01294 | HMTase inhibitor
RG 108 | DNA methylation inh.
YS 49 | antithrombotic
MDL 201012 | M3 antagonist
STF 083010 | IRE1 inhibitor
PF 02341066 | c-Met/ALK inh.
2011 AUG
KU 55933 | ATM inhibitor
LY 317615 | PKCβ inhibitor
GSK 461364 | PLK1 inhibitor
CYT 387 | JAK1/2 inhibitor
Asoprisnil | PR modulator
RU 58841 | Antiandrogen
AEE 788 | EGFR/VEGFR inhibitor
MK 2206 | AKT inhibitor
Y-27632 | ROCK inhibitor
2011 JULY
R 406 | Syk inhibitor
BAY 73-4506 | RTK inhibitor
BINA | mGluR2 PAM
Danoprevir | HCV protease inh.
PD 173074 | FGFR inhibitor
TWS 119 | GSK-3β inhibitor
SCIO 469 | p38 MAPK inhibitor
See more ligands in 2011
2012: NEW MAR FEB JAN; 2011: DEC NOV OCT SEP AUG JULY JUN MAY APR MAR FEB JAN; 2010 2009
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