JNJ 63533054

Based on 5 reference(s) in Google Scholar 9 10 5

Axon 2569

CAS [1802326-66-4]

MF C17H17ClN2O2
MW 316.78

  • Purity: 99%
  • Optical purity: Optically pure
  • Soluble in DMSO

JNJ 63533054

Description

Potent, brain-penetrant, orally active, and selective agonist of hGPR139 (EC50 value 16 nM; 138% of max) with no inhibitory effect on CYP450. A useful tool for exploring GPR139 pharmacology, especially when combined with NCRW0005-F05 (Axon 2609), the first potent GPR139 antagonist available.

KEYWORDS: JNJ 63533054 | supplier | GPR139 agonist | JNJ63533054 | CAS [1802326-66-4] | GPR139 | Agonist | GPCR | orphan | CNS | diabetes | metabolic | brain | tool | central nervous system

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Size Unit Price Stock
10 mg €90.00 In Stock
50 mg €310.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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