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Compound 120 

Deuterated Atazanivir

 

 

CAS 1092540-56-1

 C39H37D15N6O7.H2SO4 

Purity: 99 % (optically pure)

Soluble in DMSO to 59 mM

 

 

 

 

 

Ordering Information:

 

Cat. No. Axon 1753     Exclusive Promotion

 

Qty1: 2 mg (research sample) / 115  $150

 

Qty2: 5 mg (research sample) / €175  $228

 

Qty3: on request

 

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or by fax to: +31-50-3600390.

 

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Biological Activity:

 

A partially deuterated analog of Atazanivir (Axon 1441), an oral HIV protease inhibitor; A deuterium-containing medicine with improved ADME properties; Compound 120 showed an approximately 50% increase in half life compared with Atazanavir.

 

References: online

 

 

 

 

 

Chemical Name: 

 

Deuterated Atazanivir | Protease inhibitor | Axon Medchem | Axon 1753 | Compound 120

 

Axon Ligands TM - Research chemicals for biological study. Some high-profile samples could be provided under terms of contract research synthesis.

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Axon Ligands in the field:

 

AG 7088 | HRV 3C inhibitor

Atazanivir | Protease inhibitor

D-Atazanivir | Protease inhibitor

Danoprevir | HCV protease inh.

Nelfinavir | Protease inhibitor

Dapivirine | NNRT inhibitor