Axon Ligands (TM) - alphabetic: [A] [B] [C] [D] [E] [F] [G] [H] [I] [J] [K] [L] [M] [N] [O] [P] [Q] [R] [S] [T] [U] [V] [W] [X] [Y] [Z]

SB 242084 dihydrochloride

CAS 1049747-87-6

181632-25-7 (free base)

C21H19ClN4O2.2HCl  MW 467.78

Purity: 99%

Soluble in water and DMSO

Ordering Information:

Cat. No. Axon 1745   Prime Source 

Qty1: 5 mg / €115  $150

Qty2: 25 mg / €415  $540

Qty3: on request

Send enquiry to: order@axonmedchem.com

or by fax to: +31-50-3600390.

Contact us for payment and tech support.

Biological Activity:   Selective and brian penetrant 5-HT2C receptor antagonist   References: online   SM Bromidge et al. 6-Chloro-5-methyl-1-[[(2-methyl-3-pyridyl)oxy]-5-pyridyl]carbamoyl]-indoline (SB-242084): the first selective and brain penetrant 5-HT2C receptor antagonist. J. Med. Chem. 1997, 40(22), 3494-3496. [online]   GA Kennet et al. SB 242084, a selective and brain penetrant 5-HT2C receptor antagonist. Neuropharmacology 1997, 36(4-5), 609-620. [online]   GL Dalton et al. Serotonin 1B and 2C receptor interactions in the modulation of feeding behaviour in the mouse. Psychopharmacol. 2006, 185(1), 45-57. [online]       Chemical Name: 6-chloro-5-methyl-N-(6-(2-methylpyridin-3-yloxy)pyridin-3-yl)indoline-1-carboxamide dihydrochloride

SB 242084 | 5-HT2C antagonist | Axon Medchem | Axon 1745 | SB242084

Axon Ligands TM - Research chemicals for biological study. Some high-profile samples could be provided under terms of contract research synthesis.

axonmedchem.com © 2011