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D 106669

Based on 20 reference(s) in Google Scholar 80 100 20

Axon 1719

CAS [938444-93-0]

MF C17H18N6O
MW 322.36

  • Purity: 98%
  • Soluble in DMSO

D 106669

Description

Highly potent and selective PI3K inhibitor, selectively inhibiting class I PI3K (PI3Kα IC50 <10 nM, >3 log selectivity against tyrosine or serine/threonine kinases, except ERK1 and 2) and showed some activity in A549 (lung cancer) xenografts mouse model at oral dose of 30 mg/kg twice daily
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Size Unit Price Stock
2 mg €85.00 In Stock
5 mg €120.00 In Stock
25 mg €420.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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