GSK 3787 | PPAR δ antgonist | Axon Medchem | Axon 1628

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GSK 3787

CAS 188591-46-0

C15H12ClF3N2O3S MW 392.78

Purity: 99%

Soluble in DMSO (32 mg/mL)

Ordering Information:

Cat. No. Axon 1628 Prime Source Promotion

Qty1: 10 mg / €115 $150

Qty2: 50 mg / €415 $540

Qty3: on request

Send enquiry to: order@axonmedchem.com

or by fax to: +31-50-3600390.

Biological Activity:

Selective and irreversible peroxisome proliferator-activated receptor (PPAR) delta (PPARδ) antagonist.

References:

PS Palkar et al. Cellular and Pharmacological Selectivity of the PPARβ/δ Antagonist GSK3787. Mol. Pharmacol. Fast Forward. 2010.06.01. [online]

BG Shearer et al. Identification and characterization of 4-chloro-N-(2-{[5-trifluoromethyl)-2-pyridyl]sulfonyl}ethyl)benzamide (GSK3787), a selective and irreversible peroxisome proliferator-activated receptor delta (PPARdelta) antagonist. J. Med. Chem. 2010, 53(4), 1857-61. [online]

Chemical Name: 4-Chloro-N-[2-[[5-(trifluoromethyl)-2-pyridinyl]sulfonyl]ethyl]benzamide

GSK 3787 | PPAR δ antgonist | Axon Medchem | Axon 1628 | GSK3787

Axon Ligands ^TM - Research chemicals for biological study. Some high-profile samples could be provided under terms of contract research synthesis.

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