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CID 755673

 

 

CAS 521937-07-5

C12H11NO3  MW 217.22

Purity: >98%

Soluble in DMSO (40 mg/mL)

 

 

 

 

Ordering Information:

 

Cat. No. Axon 1627    

 

Qty1: 10 mg / €125  $163

 

Qty3: 50 mg / €425  $553

 

Qty4: on request

 

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Biological Activity:

 

Selective protein kinase D (PKD) inhibitor

 

References:

 

ER Sharlow et al. Potent and Selective Disruption of Protein Kinase D Functionality by a Benzoxoloazepinolone. J. Biol. Chem. 2008, 283, 33516-33526. [online]

 

E Torres-Marquez et al. CID755673 enhances mitogenic signaling by phorbol esters, bombesin and EGF through a protein kinase D-independent pathway.
Biochem. Biophys. Res. Commun. 2010, 391(1), 63-68. [online]

 

 

Chemical Name: 7-Hydroxy-2,3,4,5-tetrahydro-1H-[1]benzofuro[2,3-c]azepin-1-one

 

CID 755673 | PKD inhibitor | Axon Medchem | Axon 1627 | CID755673

Axon Ligands TM - Research chemicals for biological study. Some high-profile samples could be provided under terms of contract research synthesis.

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Axon Ligands In The Field:

 

CID 755673 | PKD inhibitor

 

AEB 071 | PKC inhibitor

LY 317615 | PKCβ inhibitor

LY 333531 | PKCβ inhibitor

 

 

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