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MK 0354

CAS 851776-28-8

C7H8N6  MW 176.18

Purity: 99%

Soluble in DMSO

Ordering Information:

Cat. No. Axon 1576    Prime Source Promotion

Qty1: 10 mg / €135  $176

Qty2: 50 mg / €535  $696

Qty3: on request

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Biological Activity:   Partial agonist of Naicin receptor, GPR109a.   References:   E Lai et al, Effects of a niacin receptor partial agonist, MK-0354, on plasma free fatty acids, lipids, and cutaneous flushing in humans. J. Clin. Lipidol. 2008, 2(5), 375-383. [online]   G Semple et al. 3-(1H-tetrazol-5-yl)-1,4,5,6-tetrahydro-cyclopentapyrazole (MK-0354): a partial agonist of the nicotinic acid receptor, G-protein coupled receptor 109a, with antilipolytic but no vasodilatory activity in mice. J. Med. Chem. 2008, 51(16), 5101-5108. [online]     Chemical Name: 3-(1H-tetrazol-5-yl)-1,4,5,6-tetrahydro-cyclopentapyrazole

MK 0354 | Niacin receptor partial agonist | Axon Medchem | Axon 1576 | MK0354

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Axon Ligands In The Field:

MK 0354 | Naicin partial agonist