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AR 231453

 

 

CAS 733750-99-7

C21H24FN7O5S MW 505.5

Purity: 99%

 

 

 

 

Ordering Information:

 

Cat. No. Axon 1572   Prime Source Promotion

 

Qty1: 5 mg (reseach sample) / €95  $124

 

Qty2: 25 mg (research sample) / €285  $371

 

Qty3: on request contract research synthesis

 

Send enquiry to: order@axonmedchem.com

or by fax to: +31-50-3600390.

 

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Biological Activity:  

 

Potent and orally active agonist of cannabinoid receptor GPR119.

 

References: online

 

G Semple et al. Discovery of the first potent and orally efficacious agonist of the orphan G-protein coupled receptor 119. J Med Chem. 2008, 51(17), 5172–5175.

 

 

 

Chemical Name: N-(2-fluoro-4-methanesulfonylphenyl)-(6-[4-(3-isopropyl-[1,2,4]oxadiazol-5-yl)-piperidin-1-yl]-5-nitro-pyrimidin-4-yl)amine

 

AR 231453 | GPR119 agonist | Axon Medchem | Axon 1572 | AR231453

Axon Ligands TM - Research chemicals for biological study. Some high-profile samples could be provided under terms of contract research synthesis.

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Axon Ligands In The Field:

 

AR 231453 | GPR119 agonist

Palmitoylethanolamide | GPR55 agonist

 

Abn-CBD | Axon 1235

Cannabidiol - CBD | Axon 1234

HU-308 | CB2 agonist

Iodopravadoline | CB antagonist

JWH 018 | CB2 agonist

JWH 073 | CB2 agonist 

JWH 133 | CB2 agonist

JWH 250 | CB agonist

Pravadoline | CB agonist

AM 251 | CB1 antagonist

AM 281 | CB1 antagonist

PSNCBAM-1 | CB1 antagonist

SR 141716 | CB1 antagonist