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GSK 650394

CAS 890842-28-1

C25H22N2O2  MW 382.45

Purity: 99%

Ordering Information:

Cat. No. Axon 1570   Prime Source

Qty1:  5 mg (research sample) / €95  $124

Qty2: 10 mg (research sample) / €135  $176

Qty3: 25 mg (research sample) / inquire 

Qty4: on request

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Biological Activity:   Specific inhibitor of serum- and glucocorticoid-regulated kinases 1 (SGK 1), with IC50 values to be 62 and 103 nM for SGK1 and SGK2 respectively.    References:   AB Sherk et al. Development of a small molecule serum and glucocorticoid-regulated kinase 1 antagonist and its evaluation as a prostate cancer therapeutic. Cancer Res. 2008, 68(18), 7475–7483. [online]     Chemical Name: 2-Cyclopentyl-4-(5-phenyl-1H-pyrrolo[2,3-b]pyridin-3-yl-benzoic acid

GSK 650394 | SGK inhibitor | Axon Medchem | Axon 1570 | GSK650394

Axon Ligands In The Field:

GSK 650394 | SGK inhibitor