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PSNCBAM-1

CAS 877202-74-9

C22H21ClN4O MW 392.89

Purity: 99 %

Ordering Information:

Cat. No. Axon 1565   Prime Source

Qty1: 5 mg (research sample) / €105  $137 

Promotion: 2 x 5 mg / €150  $195 

Qty2: 25 mg (research sample) / €350  $455 

Promotion: 2 x 25 mg / €520  $676 

Qty3: on request

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Biological Activity:   An allosteric CB1 receptor antagonist, potentially an anti-obesity agents.   References:   JG Horswill et al. PSNCBAM-1, a novel allosteric antagonist at cannabinoid CB1 receptors with hypophagic effects in rats. Br J Pharmacol. 2007, 152(5), 565-6. [online]   JG Horswill et al. Characterisation of PSNCBAM-1, a novel allosteric antagonist of the cannabinoid type 1 receptor with in vivo efficacy in an acute rat feeding model. PBPS 2006. [abstract]       Chemical Name: 1-(2,4-Dichloro-phenyl)-5-(4-iodo-phenyl)-4-methyl-1H-pyrazole-3-carboxylic acid piperidin-1-ylamide

PSNCBAM-1 | CB1 antagonist | Axon Medchem | Axon 1565

Axon Ligands TM - Research chemicals for biological study. Some high-profile samples could be provided under terms of contract research synthesis.

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