Droperidol | D2 antagonist | Axon Medchem

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Droperidol

R 4749 - Droleptan - Dridol

CAS 548-73-2

C22H22FN3O2 MW 379.43

Purity: 99 %

Ordering Information:

Cat. No. Axon 1554

Qty1: 100 mg / 105 $137

Qty2: 500 mg / 405 $527

Qty3: on request

Send enquiry to: order@axonmedchem.com

or by fax to: +31-50-3600390.

Biological Activity:

Dopamine D2 receptor antagonist and α1 adrenoceptor antagonist; an antidopaminergic drug used as an antiemetic and antipsychotic; also often used for neuroleptanalgesic anesthesia and sedation in intensive-care treatment.

References: online

S Purhonen et al. Comparison of tropisetron, droperidol, and saline in the prevention of postoperative nausea and vomiting after gynecologic surgery. Anesth Analg 1997, 84(3), 662-667. [online]

SJ Wang et al. Droperidol treatment of status migrainosus and refractory migraine. Headache 1997, 37(6), 377-382. [online]

M Koivuranta et al. The antiemetic efficacy of a combination of ondansetron and droperidol. Anaesthesia 1997, 52(9), 863-868. [online]

Chemical Name: 1-{1-[4-(4-Fluoro-phenyl)-4-oxo-butyl]-1,2,3,6-tetrahydro-pyridin-4-yl}-1,3-dihydro-benzoimidazol-2-one

Droperidol | D2 antagonist | Axon Medchem | Axon 1554