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Axon Ligands (TM) - alphabetic: [A] [B] [C] [D] [E] [F] [G] [H] [I] [J] [K] [L] [M] [N] [O] [P] [Q] [R] [S] [T] [U] [V] [W] [X] [Y] [Z]

 

 

 

  

Pravadoline - WIN 48098

 

CAS 92623-83-1

C23H26N2O3  MW 378.48

Purity: 99%

 

 

 

 

Ordering Information:

 

Cat. No. Axon 1523    

 

Qty1: 10 mg / €105  $137

 

Qty2: 50 mg / €315  $410

 

Qty3: on request

 

Send enquiry to: order@axonmedchem.com

or by fax to: +31-50-3600390.

 

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Biological Activity:

 

COX inhibitor and cannabinoid (CB) agonist, an antiinflammatory and analgesic agent.

 

References: online

 

DR Haubrich, et al. Pharmacology of pravadoline: a new analgesic agent. J. Pharmacol. Exp. Ther. 1990, 255(2), 511–522.

 

TE D'Ambra et al. Conformationally restrained analogues of pravadoline: nanomolar potent, enantioselective, (aminoalkyl)indole agonists of the cannabinoid receptor. J. Med. Chem. 1992, 35(1), 124–135.

 

 

Chemical Name: (4-methoxyphenyl)-[2-methyl-1-(2-morpholin-4-ylethyl)indol-3-yl]methanone

 

Pravadoline | COX inhibitor, CB agonist | Axon Medchem | Axon 1523

axonmedchem.com © 2010

 

Axon Ligands In The Field:

 

Abn-CBD | Axon 1235

Cannabidiol - CBD | Axon 1234

HU-308 | CB2 agonist

Iodopravadoline | CB antagonist

JWH 018 | CB2 agonist

JWH 073 | CB2 agonist 

JWH 133 | CB2 agonist

JWH 250 | CB agonist

Pravadoline | CB agonist

AM 251 | CB1 antagonist

AM 281 | CB1 antagonist

MK 0364 | CB1 inverse agonist

PSNCBAM-1 | CB1 antagonist

SR 141716 | CB1 antagonist