Aprepitant

Based on 20 reference(s) in Google Scholar 80 100 20

Axon 1486

CAS [170729-80-3]

MF C23H21F7N4O3
MW 534.43

Purity: 99%
Optical purity: Optically pure
Soluble in DMSO

Aprepitant

Description

Substance P antagonist (SPA), having effect by blocking the neurokinin 1 (NK1) receptor

K Ranga and R Krishnan. Clinical experience with substance P receptor (NK1) antagonists in depression. J. Clin. Psychiatry 2002, 63 Suppl 11, 25-9.

AK Majumdar et al. Effects of aprepitant on cytochrome P450 3A4 activity using midazolam as a probe. Clin. Pharmacol. Ther. 2003, 74, 150–156.

CNS Pain & Inflammation A9 Tachykinin (NK)

Substance P antagonist (SPA); NK1 inhibitor

Chemical name

5-[(2R,3S)-2-[(R)-1-(3,5-Bis-trifluoromethyl-phenyl)-ethoxy]-3-(4-fluoro-phenyl)-morpholin-4-ylmethyl]-2,4-dihydro-[1,2,4]triazol-3-one

Parent CAS No.

[170729-80-3]

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