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Risperidone

R 64766

 

CAS 106266-06-2

C23H27FN4O2  MW 410.48

Purity: 99%

 

 

 

 

Ordering Information:

 

Cat. No. Axon 1454

 

Qty1: 10 mg / 85  $111

 

Qty2: 50 mg / 255  $332

 

Qty3: on request

 

Send enquiry to: order@axonmedchem.com

or by fax to: +31-50-3600390.

 

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Biological Activity:

 

5-HT2 and dopamine D2 antagonist with high affinity for 5-HT7 receptors; an atypical antipsychotic in the treatment of psychotic disorders with negative and positive symptomatology.

 

References: online

 

Leysen et al. Biochemical profile of risperidone, a new antipsychotic. J. Pharmacol. Exp. Ther. 1988, 247, 661.

 

Stathis et al. Risperidone: a novel antipsychotic with many "atypical" properties. Psychopharmacol. 1996, 127, 181.

 

A Szarfman et al. Atypical antipsychotics and pituitary tumors: a pharmacovigilance study. Pharmacotherapy 2006, 26(6), 748–58. [abstract]

 

 

 

Chemical Name: 3-[2-[4-(6-Fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl] ethyl]-6,7,8,9-tetrahydro-2-methyl-4H-pyrido[1,2-a]pyri midin-4-one

Risperidone | Atypical antipsychotic | Axon Medchem | Axon 1454 | R 64766 - Risperidal

Axon LigandsTM

Research chemicals for biological study. Some high-profile samples could be provided under terms of contract research synthesis.

axonmedchem.com © 2010

 

Axon Atypical Antipsychotics available: e.g.

 

Amisulpride (Axon 1381)

Aripiprazole (Axon 1143)

Asenapine (Axon 1503)

Bifeprunox (Axon 1508)

Clozapine (Axon 1146)

GMC 1-169 (Axon 1148)

GMC 2-83 (Axon 1150)

GMC 61-39 (Axon 1149)

Iloperidone (Axon 1493)

Olanzapine (Axon 1298)

Quetiapine (Axon 1354)

Risperidone (Axon 1454)

Sertindole (Axon 1141)

Thio-aripiprazole (Axon 1144)

Ziprasidone (Axon 1446)

 

"Typical Antipsychotic":

Isoclozapine (Axon 1147)

 

Clozapine Analogues:

GMC 1-116 (Axon 1151)

GMC 1-165 (Axon 1152)