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Ketanserin - R 41468

CAS 74050-98-9
C22H22FN3O3  MW 395.43 

Purity: 99%

Ordering Information:

Cat. No. Axon 1450     

Qty1: 10 mg / €55  $72

Qty2: 50 mg / €95  $124

Qty3: on request

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Biological Activity:     5-HT2A receptor antagonist; an antihypertensive; with tritium (3H) radioactively labeled ketanserin is used as a radioligand for the serotonin 5-HT2A receptor, e.g. in receptor binding assays and autoradiography.   References: online   A. Pazos et al. Serotonin receptors in the Human Brain—IV. Autoradiographic mapping of serotonin-2 receptors. Neuroscience 1987, 21(1), 123–139. [abstract] L Sharon et al.. Expression of serotonin 5-HT2A receptors in the human cerebellum and alterations in schizophrenia. Synapse 2001, 42(2), 104–114. [abstract]      Chemical Name: 3-[2-[4-(4-Fluorobenzoyl)-1-piperidinyl]ethyl]-2,4[1H,3 H]-quinazolinedione

Ketanserin | 5-HT2A antgonist | Axon Medchem | Axon 1450 | R 41468

Axon Ligands TM - Research chemicals for biological study. Some high-profile samples could be provided under terms of contract research synthesis.

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Axon Ligands In The Field:

Risperidon | 5-HT2A antagonist

Ziprasidone | 5-HT2/D2 antag.